Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_00221
Ion Channel
ATP-sensitive inward rectifier potassium channel 10
Peptide Function
Blocker
Gene Name
KCNJ10
Activity Data (nM)
IC50
100 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
ALCNCNRIIIPHQCWKKCGKK
Peptide UniProt Accession
UniParc
UPI0000D6EB06
Peptide Synonyms/Alias
[Tertiapin Q; Tertiapin Q [MI]; UNII-2KDS4KK188; 2KDS4KK188; EX-A7698; Ala-leu-cys-asn-cys-asn-arg-ile-ile-ile-pro-his-gln-cys-trp-lys-lys-cys-gly-lys-lys]
Peptide Species
Apis mellifera (Honeybee)
Peptide Name
Tertiapin
CAS Number
Not available
Experimental Conditions
pH
pH 7.4
Holding Potential (mV)
−80 to 80 mV
Temperature
Room Temperture
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
Kir
Ion Channel UniProt Accession
Source Organism
Mus musculus (Mouse)
References & Disease Information
Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available